Targeting reward-relevant nicotinic receptors in the discovery of novel pharmacotherapeutic agents to treat tobacco dependence

Nebr Symp Motiv. 2009:55:31-63. doi: 10.1007/978-0-387-78748-0_4.
No abstract available

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Animals
  • Benzazepines / adverse effects
  • Benzazepines / therapeutic use
  • Brain / drug effects
  • Brain / physiopathology
  • Bupropion / adverse effects
  • Bupropion / therapeutic use
  • Dopamine / metabolism
  • Dose-Response Relationship, Drug
  • Drugs, Investigational / adverse effects
  • Drugs, Investigational / pharmacology
  • Drugs, Investigational / therapeutic use*
  • Male
  • Neurons / drug effects
  • Neurons / physiology
  • Nicotine / adverse effects
  • Nicotine / therapeutic use
  • Nicotinic Antagonists / adverse effects
  • Nicotinic Antagonists / pharmacology
  • Nicotinic Antagonists / therapeutic use*
  • Picolines / adverse effects
  • Picolines / pharmacology
  • Picolines / therapeutic use
  • Quaternary Ammonium Compounds / adverse effects
  • Quaternary Ammonium Compounds / pharmacology
  • Quaternary Ammonium Compounds / therapeutic use
  • Quinoxalines / adverse effects
  • Quinoxalines / therapeutic use
  • Rats
  • Rats, Inbred F344
  • Rats, Sprague-Dawley
  • Receptors, Nicotinic / drug effects*
  • Receptors, Nicotinic / physiology
  • Reward*
  • Smoking Cessation / psychology*
  • Structure-Activity Relationship
  • Tobacco Use Disorder / physiopathology
  • Tobacco Use Disorder / rehabilitation*
  • Varenicline
  • Ventral Tegmental Area / drug effects
  • Ventral Tegmental Area / physiology
  • alpha7 Nicotinic Acetylcholine Receptor

Substances

  • Benzazepines
  • Chrna7 protein, rat
  • Drugs, Investigational
  • N,N'-dodecane-1,12-diyl-bis-3-picolinium dibromide
  • Nicotinic Antagonists
  • Picolines
  • Quaternary Ammonium Compounds
  • Quinoxalines
  • Receptors, Nicotinic
  • alpha7 Nicotinic Acetylcholine Receptor
  • Bupropion
  • Nicotine
  • Dopamine
  • Varenicline